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Regioselective Enzymatic Acylation of Aureolic Acids to Obtain Novel Analogues with Improved Antitumor Activity

Author:
González Sabín, JavierUniovi authority; Núñez González, Luz ElenaUniovi authority; Fernández Braña, Alfredo JavierUniovi authority; Méndez Fernández, María del CarmenUniovi authority; Salas Fernández, José AntonioUniovi authority; Gotor Santamaría, Vicente MiguelUniovi authority; Morís Varas, Francisco
Publication date:
2012
Publisher version:
http://dx.doi.org/10.1002/adsc.201100944
Citación:
Advanced Synthesis & Catalysis, 354, p. 1500–1508 (2012); doi:10.1002/adsc.201100944
URI:
http://hdl.handle.net/10651/9032
ISSN:
1615-4169
Identificador local:

20120720

DOI:
10.1002/adsc.201100944
Patrocinado por:

We thank M. A. Hermosilla and M. L. Aller for assistance inthe enzyme screening and product purifications. We are alsogratefully acknowledged the National Cancer Institute (Be-thesda, MD) for the antitumor assays.

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