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Discovery of Reversible DNA Methyltransferase and Lysine Methyltransferase G9a Inhibitors with Antitumoral in Vivo Efficacy

dc.contributor.authorRabal, O.
dc.contributor.authorJosé Enériz, E. S.
dc.contributor.authorAguirre, Xabier
dc.contributor.authorFernández Fraga, Mario 
dc.date.accessioned2018-11-27T08:03:52Z
dc.date.available2018-11-27T08:03:52Z
dc.date.issued2018
dc.identifier.citationJournal of Medicinal Chemistry, 61(15), p. 6518-6545 (2018); doi:10.1021/acs.jmedchem.7b01926
dc.identifier.issn0022-2623
dc.identifier.urihttp://hdl.handle.net/10651/49408
dc.description.sponsorshipFoundation for Applied Medical Research (FIMA); Fundacion Fuentes Dutor; Ministerio de Economia y Competitividad; Instituto de Salud Carlos III (FEDER funds) [PI10/01691, PI13/00862, PI13/01469, PI14/01867, PI16/02024, PI17/00701, RTICC RD12/0036/0068, CIBERONC (GB16/12/00489)]; ERA NET programs TRANSCAN-2 JTC EPICA by the "Torres Quevedo" Subprogram [PTQ-11-04777, PTQ-14-07320 I.D.M.]; Fundaci La Marato de TV3 [20132130-31-32]; Gobierno de Navarra [40/2016, PT053/2016, PT027/2017]; FSE (Inncorpora-Torres Quevedo grant); Plan Nacional de I+D+I 2013-2016/FEDER [PI15/00892]; Asturias Regional Government [GRUPIN14-052]; IUOPA-Obra Social Liberbank-Cajastur; University of Navarra (Pamplona, Spain); Asociacion de Amigos of University of Navarra
dc.description.statementofresponsibilityRabal, O., José-Enériz, E.S., Agirre, X., Sánchez-Arias, J.A., Vilas-Zornoza, A., Ugarte, A., De Miguel, I., Miranda, E., Garate, L., Fraga, M., Santamarina, P., Perez, R.F., Ordoñez, R., Sáez, E., Roa, S., García-Barchino, M.J., Martínez-Climent, J.A., Liu, Y., Wu, W., Xu, M., Prosper, F., Oyarzabal, J.
dc.format.extentp. 6518-6545
dc.language.isoeng
dc.relation.ispartofJournal of Medicinal Chemistry
dc.rights© 2018 American Chemical Society
dc.sourceScopus
dc.source.urihttps://www.scopus.com/inward/record.uri?eid=2-s2.0-85049372799&doi=10.1021%2facs.jmedchem.7b01926&partnerID=40&md5=5b88adf8e3e37cdd8b2160163c803d19
dc.titleDiscovery of Reversible DNA Methyltransferase and Lysine Methyltransferase G9a Inhibitors with Antitumoral in Vivo Efficacy
dc.typejournal article
dc.identifier.doi10.1021/acs.jmedchem.7b01926
dc.relation.projectIDPI10/01691
dc.relation.projectIDGB16/12/00489
dc.relation.projectIDPTQ-11-04777
dc.relation.publisherversionhttp://dx.doi.org/10.1021/acs.jmedchem.7b01926


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